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Home - Products - Cell Cycle/DNA Damage - GPR - PSN 375963

PSN 375963

CAS No. 388575-52-8

PSN 375963( PSN 375963 hydrochloride | PSN 375963 )

Catalog No. M27691 CAS No. 388575-52-8

PSN 375963 hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 36 Get Quote
5MG 58 Get Quote
10MG 88 Get Quote
25MG 177 Get Quote
50MG 295 Get Quote
100MG 484 Get Quote
200MG 690 Get Quote
500MG 1035 Get Quote
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Biological Information

  • Product Name
    PSN 375963
  • Note
    Research use only, not for human use.
  • Brief Description
    PSN 375963 hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.
  • Description
    PSN 375963 hydrochloride is a synthetic agonist of the endogenous ligand for GPR119.(In Vitro):PSN 375963 is a potent GPR119 agonist with EC50s of 8.4 and 7.9 μM for human and mouse GPR119.(In Vivo):PSN 375963 suppressed food intake in rats and reduced body weight gain and white adipose tissue deposition upon subchronic oral administration to high-fat-fed rats.
  • In Vitro
    The endogenous ligand OEA signals through GPR119 in a manner similar to glucagon-like peptide-1 (GLP-1) and its receptor with respect to insulin secretion, intracellular calcium and cAMP.
  • In Vivo
    ——
  • Synonyms
    PSN 375963 hydrochloride | PSN 375963
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    GPR
  • Recptor
    NDM-1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    388575-52-8
  • Formula Weight
    321.85
  • Molecular Formula
    C17H24ClN3O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 50 mg/mL (175.20 mM)
  • SMILES
    Cl.CCCC[C@H]1CC[C@@H](CC1)c1nc(no1)-c1ccncc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Cui-Gai Bai, et al. Cysteine and Its Derivatives as New Delhi Metallo-beta-lactamase-1 Inhibitors. Current Enzyme Inhibition, 2015, 11, 46-57
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